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  Drug Discovery ½ÉÆ÷Áö¿ò ¹× ±³À° ¾È³»
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ÀúÈñ ºÐÀÚ¼³°è¿¬±¸¼Ò(Research Institute of Bioinformatics & Molecular Design)´Â ÄÄÇ»Å͸¦ ÀÌ¿ëÇÏ¿© »ý¹°/È­ÇÐ Á¤º¸ÇÐ ¹× ½Å¾à/½Å¼ÒÀç °³¹ßÀ» ¿¬±¸ÇÏ´Â °÷À¸·Î ¸Å³â ½Å¾à°³¹ß±³À°À» ½Ç½ÃÇÏ°í ÀÖ½À´Ï´Ù.  2004³â ½Ç½ÃµÇ´Â ½Å¾à±³À°Àº Á¾Àü±³À°°ú´Â Â÷º°È­µÈ ¹æ¹ýÀ¸·Î °³ÃÖµÉ ¿¹Á¤ÀÔ´Ï´Ù.  ù°³¯ ½Å¾à°ü·Ã ±¹³»¿Ü Àú¸íÇÐÀÚµéÀ» ÃʺùÇÏ¿© ½ÉÆ÷Áö¿òÀ» °³ÃÖÇÑ ÈÄ Ã¹Â°³¯ ¿ÀÈĺÎÅÍ µÑ°³¯±îÁö Àü¹®°¡±³À°À» ½Ç½ÃÇÕ´Ï´Ù.  ÀÌ Àü¹®°¡±³À°Àº ½ÉÆ÷Áö¿ò ÈÄ Á» ´õ ÀÚ¼¼ÇÑ ³»¿ëÀ¸·Î ÀÌ·ÐÀ§ÁÖÀÇ ±³À°À» ½Ç½ÃÇÒ °ÍÀÔ´Ï´Ù. ¼Â°³¯°ú ³Ý°³¯Àº ¾ÕÀÇ ½ÉÆ÷Áö¿ò°ú Àü¹®°¡ ±³À°À» Åä´ë·Î Á÷Á¢ ½Ç½ÀÀ» ÇÏ¿© ±³À°³»¿ëÀ» ¿ÏÀüÈ÷ ½ÀµæÇÏ¿© Project¿¡ Àû¿ë ÇÒ ¼ö ÀÖµµ·Ï ÁøÇàµÉ ¿¹Á¤ÀÔ´Ï´Ù.  °ü½É ÀÖ´Â ºÐµéÀÇ ¸¹Àº Âü¿©¹Ù¶ø´Ï´Ù.

1. Structural Bio & Cheminformatics for Drug Discovery Symposium
- ³¯ Â¥ : 2004³â 8¿ù 24ÀÏ (È­)
- Àå ¼Ò : ¿¬¼¼´ëÇб³ ¿¬¼¼°øÇпø ÁöÇÏ1Ãþ ´ë°­´ç
- µî ·Ï ºñ : 2¸¸¿ø
- ÇÁ·Î±×·¥
* X-ray¸¦ ÀÌ¿ëÇÑ Structure Based Drug Design- Å©¸¯½ºÅ»Áö³ë¹Í½º(ÁÖ)
* A computational pipeline for protein structure prediction and analysis at genome scale - ±èµ¿¼· ±³¼ö (KAIST)
* Discovering Leads Using Virtual Screening - Prof. HualIang Jiang (Shanghai Institute of Materia Medica, CHINA)
* Virtual Screening Case Studies Using LigandFit - Dr. Hongwei Huang (Accelrys K.K., Tokyo, JAPAN)
* Developing Virtual Screening Program for Lead Identification - ³²±â¿± ¹Ú»ç (BMD)
* in silico Lead Generation - (ÁÖ)¾ÆÀ̵ð¾Ë

2. ½Å¾à °³¹ß ±³À°
(1) Àü¹®°¡ ±³À°
 - °­Á¸í : Structural Bio & Cheminformatics for Drug Discovery
 - ³¯ Â¥ : 8¿ù 24ÀÏ ~ 25ÀÏ
 - Àå ¼Ò : ¿¬¼¼´ëÇб³ ¿¬¼¼°øÇпø 2Ãþ ¼¼¹Ì³ª½Ç
 - ¼ö°­·á : 10¸¸¿ø (½ÉÆ÷Áö¿ò µî·Ïºñ Æ÷ÇÔ)
 - ¼ö°­Àοø : ¾à 40¸í
 - ÇÁ·Î±×·¥
 * Introduction to CADD - ³ë°æÅÂ(BMD)
 * ab initio Protein Structure Prediction for Target Protein - Á¶±¤ÈÖ(¼þ½Ç´ë)
 * Target Protein Structure Prediction by Threading technology - ±èµ¿¼·(KAIST)
 * Homology Modeling for Target Protein Modeling - ±è³²µÎ(IDR)
 * Introduction to Cheminformatics - À庴ÇÏ(IDR)
 * Ligand Docking for Drug Discovery - ³²±â¿±(BMD)
 * Virtual Screening for Lead Identification - À±Á¤Çõ(IDR)

(2) Extensive Course
 - ³¯ Â¥ : 8¿ù 26ÀÏ ~ 27ÀÏ (2ÀÏ)
 - Àå ¼Ò : (»ç)ºÐÀÚ¼³°è¿¬±¸¼Ò ¿¬±¸½Ç
 - ¼ö°­·á : 100¸¸¿ø
 - ¼ö°­Àοø : ¾à 10¸í(¼±Âø¼ø)

¡Ø º» ±³À°Àº ¼ö°­ÀÚ À§ÁÖÀÇ ¸ÂÃã ±³À°ÀÔ´Ï´Ù.
(»ç)ºÐÀÚ¼³°è¿¬±¸¼Ò¿Í (ÁÖ)¾ÆÀ̵ð¾Ë¿¡¼­´Â °¢ ¿¬±¸ ´Ü°èº° ÃÊÁ¡À» ¸ÂÃá ´Ù¾çÇÑ ¿¬±¸»ç·Ê¸¦ ±³À° ¹ÞÀ» ¼ö ÀÖ´Â ±âȸ¸¦ Á¦°øÇÕ´Ï´Ù.

´ÙÀ½ÀÇ ±âº»ÀûÀÎ 4´Ü°è°¡ ±âº» Ä¿¸®Å§·³À̸ç, ±× ¿Ü ÇÊ¿ä ¿äû½Ã Ãß°¡±³À°ÀÌ °¡´ÉÇÕ´Ï´Ù.

¨ç Protein structure Modeling
  - Homology modeling
  - Virtual screening for lead generation
¨è Docking
  - Virtual screening for lead generation
  - De novo design for lead optimization
¨é QSAR
  - Hit evaluation for lead generation
  - Lead optimization with in silico ADME/Tox. programs
¨ê Ligand Library Design
  - Virtual Combichem library design
  - Library design for lead generation

Extensive Course ½Åû ¸¶°¨Àº 8¿ù 12ÀϱîÁö À̸ç, ¼±Âø¼øÀÔ´Ï´Ù.
±³À° ½Åû½Ã ¿øÇϽô ¿¬±¸»ç·Ê¿¡ ´ëÇÏ¿© ¾Ë·Á Áֽñ⠹ٶø´Ï´Ù. (e-mail : edu@bmdrc.org)

(Extensive Course ¼ö°­·á´Â ½ÉÆ÷Áö¿ò ¹× Àü¹®°¡±³À°ºñ Æ÷ÇԱݾ×À̸ç, 1:1±³À°ÀÓ)

¡Ø µî·Ï : ȨÆäÀÌÁö¸¦ ÅëÇÑ ¿Â¶óÀεî·Ï : http://www.bmdrc.org
¡Ø ¹®ÀÇó : 02-393-9550~1 (³»¼± 204)  email : edu@bmdrc.org    http://www.bmdrc.org

   

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